5WVD
Structure of Mnk1 in complex with DS12881479
Summary for 5WVD
Entry DOI | 10.2210/pdb5wvd/pdb |
Related | 5WVJ 5WVL |
Descriptor | MAP kinase interacting serine/threonine kinase 1, SULFATE ION, 1-methyl-N-(5-phenyl-1,3-thiazol-2-yl)piperidine-4-carboxamide (3 entities in total) |
Functional Keywords | kinase, kinase inhibitor, inactive conformation, transferase |
Biological source | Homo sapiens (Human) |
Total number of polymer chains | 2 |
Total formula weight | 70189.81 |
Authors | Matsui, Y.,Hanzawa, H. (deposition date: 2016-12-24, release date: 2018-01-03, Last modification date: 2023-11-22) |
Primary citation | Matsui, Y.,Yasumatsu, I.,Yoshida, K.I.,Iimura, S.,Ikeno, Y.,Nawano, T.,Fukano, H.,Ubukata, O.,Hanzawa, H.,Tanzawa, F.,Isoyama, T. A novel inhibitor stabilizes the inactive conformation of MAPK-interacting kinase 1. Acta Crystallogr F Struct Biol Commun, 74:156-160, 2018 Cited by PubMed: 29497019DOI: 10.1107/S2053230X18002108 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (3 Å) |
Structure validation
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