5VLO
The structure of human CamKII with bound inhibitor
Summary for 5VLO
Entry DOI | 10.2210/pdb5vlo/pdb |
Descriptor | Calcium/calmodulin-dependent protein kinase type II subunit delta, N-[(2S)-2-(diethylamino)propyl]-2-[(2S)-2-(methylcarbamoyl)azetidin-1-yl]-6-[5-(thiophen-2-yl)pyrazolo[1,5-a]pyrimidin-3-yl]pyridine-4-carboxamide, 2,3-DIHYDROXY-1,4-DITHIOBUTANE, ... (4 entities in total) |
Functional Keywords | kinase, camkii, inhibitor, transferase |
Biological source | Homo sapiens (Human) |
Cellular location | Cell membrane, sarcolemma ; Peripheral membrane protein ; Cytoplasmic side : Q13557 |
Total number of polymer chains | 2 |
Total formula weight | 70321.02 |
Authors | Somoza, J.R.,Villasenor, A.G. (deposition date: 2017-04-25, release date: 2017-08-23, Last modification date: 2024-03-13) |
Primary citation | Somoza, T.J.,Villasenor, A.G. Inhibitors of CamKII To Be Published, |
Experimental method | X-RAY DIFFRACTION (2.05 Å) |
Structure validation
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