4YAY
XFEL structure of human Angiotensin Receptor
4YAY の概要
エントリーDOI | 10.2210/pdb4yay/pdb |
分子名称 | Soluble cytochrome b562,Type-1 angiotensin II receptor, 5,7-diethyl-1-{[2'-(1H-tetrazol-5-yl)biphenyl-4-yl]methyl}-3,4-dihydro-1,6-naphthyridin-2(1H)-one (2 entities in total) |
機能のキーワード | xfel, serial femtosecond crystallography, human angiotensin receptor at1r, bril, g protein-coupled receptor, gpcr, gpcr network, lipidic cubic phase, lcp, membrane protein, structural genomics, zd7155, angiotensin receptor blocker, room temperature, psi-biology |
由来する生物種 | Escherichia coli 詳細 |
タンパク質・核酸の鎖数 | 1 |
化学式量合計 | 47679.23 |
構造登録者 | Zhang, H.,Unal, H.,Gati, C.,Han, G.W.,Zatsepin, N.A.,James, D.,Wang, D.,Nelson, G.,Weierstall, U.,Messerschmidt, M.,Williams, G.J.,Boutet, S.,Yefanov, O.M.,White, T.A.,Liu, W.,Ishchenko, A.,Tirupula, K.C.,Desnoyer, R.,Sawaya, M.C.,Xu, Q.,Coe, J.,Cornrad, C.E.,Fromme, P.,Stevens, R.C.,Katritch, V.,Karnik, S.S.,Cherezov, V.,GPCR Network (GPCR) (登録日: 2015-02-18, 公開日: 2015-04-22, 最終更新日: 2023-08-16) |
主引用文献 | Zhang, H.,Unal, H.,Gati, C.,Han, G.W.,Liu, W.,Zatsepin, N.A.,James, D.,Wang, D.,Nelson, G.,Weierstall, U.,Sawaya, M.R.,Xu, Q.,Messerschmidt, M.,Williams, G.J.,Boutet, S.,Yefanov, O.M.,White, T.A.,Wang, C.,Ishchenko, A.,Tirupula, K.C.,Desnoyer, R.,Coe, J.,Conrad, C.E.,Fromme, P.,Stevens, R.C.,Katritch, V.,Karnik, S.S.,Cherezov, V. Structure of the Angiotensin receptor revealed by serial femtosecond crystallography. Cell, 161:833-844, 2015 Cited by PubMed: 25913193DOI: 10.1016/j.cell.2015.04.011 主引用文献が同じPDBエントリー |
実験手法 | X-RAY DIFFRACTION (2.9 Å) |
構造検証レポート
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