4XUM
PPARgamma ligand binding domain in complex with indomethacin
Summary for 4XUM
Entry DOI | 10.2210/pdb4xum/pdb |
Related | 4XTA 4XUH |
Descriptor | Peroxisome proliferator-activated receptor gamma, INDOMETHACIN (3 entities in total) |
Functional Keywords | ppargamma, nuclear receptor, transcription factor, nsaids, indomethacin, translation |
Biological source | Homo sapiens (Human) |
Cellular location | Nucleus: P37231 |
Total number of polymer chains | 2 |
Total formula weight | 64543.09 |
Authors | Puhl, A.C.,Webb, P.,Polikarpov, I. (deposition date: 2015-01-26, release date: 2015-11-04, Last modification date: 2024-02-28) |
Primary citation | Puhl, A.C.,Milton, F.A.,Cvoro, A.,Sieglaff, D.H.,Campos, J.C.,Bernardes, A.,Filgueira, C.S.,Lindemann, J.L.,Deng, T.,Neves, F.A.,Polikarpov, I.,Webb, P. Mechanisms of peroxisome proliferator activated receptor gamma regulation by non-steroidal anti-inflammatory drugs. Nucl Recept Signal, 13:e004-e004, 2015 Cited by PubMed: 26445566DOI: 10.1621/nrs.13004 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.4 Å) |
Structure validation
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