4U5J
C-Src in complex with Ruxolitinib
Summary for 4U5J
Entry DOI | 10.2210/pdb4u5j/pdb |
Descriptor | Proto-oncogene tyrosine-protein kinase Src, (3R)-3-cyclopentyl-3-[4-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)-1H-pyrazol-1-yl]propanenitrile (3 entities in total) |
Functional Keywords | c-src, ruxolitinib, kinase, inhibitor, transferase-transferase inhibitor complex, transferase/transferase inhibitor |
Biological source | Gallus gallus (Chicken) |
Cellular location | Cell membrane : P00523 |
Total number of polymer chains | 2 |
Total formula weight | 66066.02 |
Authors | |
Primary citation | Duan, Y.,Chen, L.,Chen, Y.,Fan, X.G. c-Src Binds to the Cancer Drug Ruxolitinib with an Active Conformation Plos One, 9:e106225-e106225, 2014 Cited by PubMed: 25197973DOI: 10.1371/journal.pone.0106225 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.26 Å) |
Structure validation
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