4PY6
Crystal Structure of bromodomain of PFA0510w from Plasmodium Falciparum
Summary for 4PY6
Entry DOI | 10.2210/pdb4py6/pdb |
Descriptor | Bromodomain protein, putative, 4-{[(7R)-8-cyclopentyl-7-ethyl-5-methyl-6-oxo-5,6,7,8-tetrahydropteridin-2-yl]amino}-3-methoxy-N-(1-methylpiperidin-4-yl)benzamide, 1,2-ETHANEDIOL, ... (4 entities in total) |
Functional Keywords | structural genomics, structural genomics consortium, sgc, bromodomain, malaria, protein binding |
Biological source | Plasmodium falciparum 3D7 |
Total number of polymer chains | 4 |
Total formula weight | 72096.21 |
Authors | Fonseca, M.,Tallant, C.,Hutchinson, A.,Savitsky, P.,Krojer, T.,Filippakopoulos, P.,Loppnau, P.,Brennan, P.E.,von Delft, F.,Dong, A.,Josling, G.A.,Duffy, M.F.,Arrowsmith, C.H.,Bountra, C.,Hui, R.,Knapp, S.,Wernimont, A.K.,Structural Genomics Consortium (SGC) (deposition date: 2014-03-26, release date: 2014-04-30, Last modification date: 2024-02-28) |
Primary citation | Fonseca, M.,Tallant, C.,Hutchinson, A.,Savitsky, P.,Krojer, T.,Filippakopoulos, P.,Loppnau, P.,Brennan, P.E.,von Delft, F.,Dong, A.,Josling, G.A.,Duffy, M.F.,Arrowsmith, C.H.,Bountra, C.,Hui, R.,Knapp, S.,Wernimont, A.K.,Structural Genomics Consortium (SGC) Crystal Structure of bromodomain of PFA0510w from Plasmodium Falciparum To be Published, |
Experimental method | X-RAY DIFFRACTION (2.5 Å) |
Structure validation
Download full validation report