4O1M
Toxoplasma gondii Enoyl acyl carrier protein reductase
Summary for 4O1M
Entry DOI | 10.2210/pdb4o1m/pdb |
Related | 2O2S 2O2Y 2O50 2PTG 3NJ8 |
Descriptor | Enoyl-acyl carrier reductase, NICOTINAMIDE-ADENINE-DINUCLEOTIDE (3 entities in total) |
Functional Keywords | rossmann fold, oxidoreductase, enoyl acyl carrier protein reductase |
Biological source | Toxoplasma gondii |
Total number of polymer chains | 6 |
Total formula weight | 204329.88 |
Authors | Muench, S.P.,Wilkinson, C.,Prigge, S.T.,Rice, D.W. (deposition date: 2013-12-16, release date: 2014-02-05, Last modification date: 2024-04-03) |
Primary citation | Wilkinson, C.,Mcphillie, M.J.,Zhou, Y.,Woods, S.,Afanador, G.A.,Rawson, S.,Khaliq, F.,Prigge, S.T.,Roberts, C.W.,Rice, D.W.,Mcleod, R.,Fishwick, C.W.,Muench, S.P. The benzimidazole based drugs show good activity against T. gondii but poor activity against its proposed enoyl reductase enzyme target Bioorg.Med.Chem.Lett., 24:911-916, 2014 Cited by PubMed: 24398298DOI: 10.1016/j.bmcl.2013.12.066 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2 Å) |
Structure validation
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