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4JVI

Crystal structure of PqsR co-inducer binding domain of Pseudomonas aeruginosa with inhibitor 3NH2-7Cl-C9QZN

Summary for 4JVI
Entry DOI10.2210/pdb4jvi/pdb
Related4JVC 4JVD
DescriptorTranscriptional regulator MvfR, 3-amino-7-chloro-2-nonylquinazolin-4(3H)-one (3 entities in total)
Functional Keywordsco-inducer binding, dna, cytoplasmic, transcription regulator-inhibitor complex, transcription regulator/inhibitor
Biological sourcePseudomonas aeruginosa
Total number of polymer chains1
Total formula weight24610.32
Authors
Ilangovan, A.,Williams, P.,Emsley, J. (deposition date: 2013-03-25, release date: 2013-08-07, Last modification date: 2024-03-20)
Primary citationIlangovan, A.,Fletcher, M.,Rampioni, G.,Pustelny, C.,Rumbaugh, K.,Heeb, S.,Camara, M.,Truman, A.,Chhabra, S.R.,Emsley, J.,Williams, P.
Structural basis for native agonist and synthetic inhibitor recognition by the Pseudomonas aeruginosa quorum sensing regulator PqsR (MvfR).
Plos Pathog., 9:e1003508-e1003508, 2013
Cited by
PubMed: 23935486
DOI: 10.1371/journal.ppat.1003508
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (2.9 Å)
Structure validation

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