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4JIN

X-ray crystal structure of Archaeoglobus fulgidus Rio1 bound to (2E)-N-benzyl-2-cyano-3-(pyridine-4-yl)acrylamide (WP1086)

Summary for 4JIN
Entry DOI10.2210/pdb4jin/pdb
Related1ZP9 1ZTF
DescriptorRIO-type serine/threonine-protein kinase Rio1, (2E)-N-benzyl-2-cyano-3-(pyridin-4-yl)prop-2-enamide (3 entities in total)
Functional Keywordsprotein kinase, ribosome biogenesis, pre-40s, autophosphorylation, transferase-transferase inhibitor complex, transferase/transferase inhibitor
Biological sourceArchaeoglobus fulgidus
Total number of polymer chains1
Total formula weight30400.95
Authors
Primary citationMielecki, M.,Krawiec, K.,Kiburu, I.,Grzelak, K.,Zagorski, W.,Kierdaszuk, B.,Kowa, K.,Fokt, I.,Szymanski, S.,Swierk, P.,Szeja, W.,Priebe, W.,Lesyng, B.,Laronde-Leblanc, N.
Development of novel molecular probes of the Rio1 atypical protein kinase.
Biochim.Biophys.Acta, 1834:1292-1301, 2013
Cited by
PubMed: 23523885
DOI: 10.1016/j.bbapap.2013.03.012
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (2.095 Å)
Structure validation

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