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4IUE

Tankyrase in complex with 7-(2-fluorophenyl)-4-methyl-1,2-dihydroquinolin-2-one

Summary for 4IUE
Entry DOI10.2210/pdb4iue/pdb
Related3W51
DescriptorTankyrase-2, ZINC ION, SULFATE ION, ... (5 entities in total)
Functional Keywordsribosylations, transferase
Biological sourceHomo sapiens (human)
Cellular locationCytoplasm: Q9H2K2
Total number of polymer chains1
Total formula weight24504.00
Authors
Jansson, A.E.,Larsson, E.A.,Nordlund, P.L. (deposition date: 2013-01-21, release date: 2013-06-26, Last modification date: 2023-11-08)
Primary citationLarsson, E.A.,Jansson, A.E.,Ng, F.M.,Then, S.W.,Panicker, R.,Liu, B.,Sangthongpitag, K.,Pendharkar, V.,Tai, S.J.,Hill, J.,Dan, C.,Ho, S.Y.,Cheong, W.W.,Poulsen, A.,Blanchard, S.,Lin, G.R.,Alam, J.,Keller, T.H.,Nordlund, P.
Fragment-based ligand design of novel potent inhibitors of tankyrases.
J.Med.Chem., 56:4497-4508, 2013
Cited by
PubMed: 23672613
DOI: 10.1021/jm400211f
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (2.38 Å)
Structure validation

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