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4IUE

Tankyrase in complex with 7-(2-fluorophenyl)-4-methyl-1,2-dihydroquinolin-2-one

Functional Information from GO Data
ChainGOidnamespacecontents
A0003950molecular_functionNAD+ poly-ADP-ribosyltransferase activity
Functional Information from PDB Data
site_idAC1
Number of Residues4
DetailsBINDING SITE FOR RESIDUE ZN A 1201
ChainResidue
ACYS1081
AHIS1084
ACYS1089
ACYS1092

site_idAC2
Number of Residues6
DetailsBINDING SITE FOR RESIDUE SO4 A 1202
ChainResidue
AHOH1341
AARG977
AHIS979
AARG980
ALYS1067
AGLN1070

site_idAC3
Number of Residues5
DetailsBINDING SITE FOR RESIDUE SO4 A 1203
ChainResidue
AASN990
AARG991
APRO1160
AGLU1161
AHOH1302

site_idAC4
Number of Residues12
DetailsBINDING SITE FOR RESIDUE AJ4 A 1204
ChainResidue
AHIS1031
AGLY1032
APRO1034
APHE1035
AHIS1048
AALA1049
ATYR1050
ATYR1060
ASER1068
ATYR1071
AILE1075
AGLU1138

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues4
DetailsBinding site: {"evidences":[{"source":"UniProtKB","id":"O95271","evidenceCode":"ECO:0000250"}]}
ChainResidueDetails

246704

PDB entries from 2025-12-24

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