4DON
Brd4 Bromodomain 1 complex with a fragment 3,4-Dihydro-3-methyl-2(1H)-quinazolinon
Summary for 4DON
Entry DOI | 10.2210/pdb4don/pdb |
Descriptor | Bromodomain-containing protein 4, 3-methyl-3,4-dihydroquinazolin-2(1H)-one (3 entities in total) |
Functional Keywords | brd4, bromodomain, four alpha helices, signaling protein |
Biological source | Homo sapiens (human) |
Total number of polymer chains | 1 |
Total formula weight | 17387.94 |
Authors | Xiong, B.,Cao, D.Y.,Chen, W.Y.,Chen, T.T.,Xu, Y.C.,Shen, J.K. (deposition date: 2012-02-09, release date: 2013-02-13, Last modification date: 2024-03-20) |
Primary citation | Xiong, B.,Cao, D.Y.,Chen, W.Y.,Chen, T.T.,Xu, Y.C.,Shen, J.K. Brd4 Bromodomain 1 complex with a fragment 3,4-Dihydro-3-methyl-2(1H)-quinazolinon To be Published, |
Experimental method | X-RAY DIFFRACTION (1.52 Å) |
Structure validation
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