4BXN
Eg5(WT) complex
Summary for 4BXN
Entry DOI | 10.2210/pdb4bxn/pdb |
Descriptor | KINESIN-LIKE PROTEIN KIF11, ADENOSINE-5'-DIPHOSPHATE, CADMIUM ION, ... (6 entities in total) |
Functional Keywords | motor protein, mitosis |
Biological source | HOMO SAPIENS (HUMAN) |
Total number of polymer chains | 2 |
Total formula weight | 86756.35 |
Authors | Talapatra, S.K.,Anthony, N.G.,Mackay, S.P.,Kozielski, F. (deposition date: 2013-07-15, release date: 2013-07-31, Last modification date: 2024-02-07) |
Primary citation | Talapatra, S.K.,Anthony, N.G.,Mackay, S.P.,Kozielski, F. The Mitotic Kinesin Eg5 Overcomes Inhibition to the Phase I/II Clinical Candidate Sb743921 by an Allosteric Resistance Mechanism. J.Med.Chem., 56:6317-, 2013 Cited by PubMed: 23875972DOI: 10.1021/JM4006274 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.793 Å) |
Structure validation
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