4BTK

TTBK1 in complex with inhibitor

Summary for 4BTK

Entry DOI	10.2210/pdb4btk/pdb
Related	4BTJ 4BTM
Descriptor	TAU-TUBULIN KINASE 1, DIMETHYL SULFOXIDE, 4-[3-HYDROXYANILINO]-6,7-DIMETHOXYQUINAZOLINE, ... (4 entities in total)
Functional Keywords	transferase, structure-kinetics relationship
Biological source	HOMO SAPIENS (HUMAN)
Cellular location	Cytoplasm : Q5TCY1
Total number of polymer chains	1
Total formula weight	39121.99
Authors	Xue, Y.,Wan, P.,Hillertz, P.,Schweikart, F.,Zhao, Y.,Wissler, L.,Dekker, N. (deposition date: 2013-06-18, release date: 2013-09-25, Last modification date: 2017-03-29)
Primary citation	Xue, Y.,Wan, P.T.,Hillertz, P.,Schweikart, F.,Zhao, Y.,Wissler, L.,Dekker, N. X-Ray Structural Analysis of Tau-Tubulin Kinase 1 and its Interactions with Small Molecular Inhibitors. Chemmedchem, 8:1846-, 2013 Cited by PubMed: 24039150 DOI: 10.1002/CMDC.201300274 PDB entries with the same primary citation
Experimental method	X-RAY DIFFRACTION (2 Å)

Structure validation