4BS6
MOUSE CATHEPSIN S WITH COVALENT LIGAND
Summary for 4BS6
Entry DOI | 10.2210/pdb4bs6/pdb |
Related | 4BQV 4BS5 4BSQ |
Descriptor | CATHEPSIN S, GLYCEROL, (2S,4R)-4-[2-chloranyl-4-(4-ethylpiperazin-1-yl)phenyl]sulfonyl-N-[1-(iminomethyl)cyclopropyl]-1-[1-(trifluoromethyl)cyclopropyl]carbonyl-pyrrolidine-2-carboxamide, ... (4 entities in total) |
Functional Keywords | hydrolase, cysteine protease, covalent ligand |
Biological source | MUS MUSCULUS (HOUSE MOUSE) |
Cellular location | Lysosome: O70370 |
Total number of polymer chains | 2 |
Total formula weight | 50625.22 |
Authors | Banner, D.W.,Benz, J.,Gsell, B.,Stihle, M.,Ruf, A.,Haap, W. (deposition date: 2013-06-07, release date: 2014-06-18, Last modification date: 2024-05-01) |
Primary citation | Haap, W.,Banner, D.W. Cathepsin S Nitrile Inhibitors To be Published, |
Experimental method | X-RAY DIFFRACTION (1.2 Å) |
Structure validation
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