4Z7I
Crystal structure of insulin regulated aminopeptidase in complex with ligand
Summary for 4Z7I
Entry DOI | 10.2210/pdb4z7i/pdb |
Descriptor | Leucyl-cystinyl aminopeptidase, DG025 transition-state analogue enzyme inhibitor, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ... (7 entities in total) |
Functional Keywords | aminopeptidase, antigen presentation, transition-state analogue, enzyme inhibitor, hydrolase, irap |
Biological source | Homo sapiens (Human) More |
Cellular location | Cell membrane ; Single-pass type II membrane protein . Leucyl-cystinyl aminopeptidase, pregnancy serum form: Secreted: Q9UIQ6 |
Total number of polymer chains | 4 |
Total formula weight | 217286.15 |
Authors | Mpakali, A.,Saridakis, E.,Harlos, K.,Zhao, Y.,Stratikos, E. (deposition date: 2015-04-07, release date: 2015-08-26, Last modification date: 2024-01-10) |
Primary citation | Mpakali, A.,Saridakis, E.,Harlos, K.,Zhao, Y.,Papakyriakou, A.,Kokkala, P.,Georgiadis, D.,Stratikos, E. Crystal Structure of Insulin-Regulated Aminopeptidase with Bound Substrate Analogue Provides Insight on Antigenic Epitope Precursor Recognition and Processing. J Immunol., 195:2842-2851, 2015 Cited by PubMed: 26259583DOI: 10.4049/jimmunol.1501103 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (3.31 Å) |
Structure validation
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