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4WF5

Crystal structure of E.Coli DsbA soaked with compound 4

Summary for 4WF5
Entry DOI10.2210/pdb4wf5/pdb
Related1FVK 4WET 4WEY 4WF4
DescriptorThiol:disulfide interchange protein, 4-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-thiazole-5-carboxylic acid, COPPER (II) ION, ... (6 entities in total)
Functional Keywordsdisulfide oxidoreductase, redox protein, dsba, oxidoreductase-oxidoreductase inhibitor complex, oxidoreductase/oxidoreductase inhibitor
Biological sourceEscherichia coli BL21(DE3)
Total number of polymer chains2
Total formula weight43102.27
Authors
Primary citationAdams, L.A.,Sharma, P.,Mohanty, B.,Ilyichova, O.V.,Mulcair, M.D.,Williams, M.L.,Gleeson, E.C.,Totsika, M.,Doak, B.C.,Caria, S.,Rimmer, K.,Horne, J.,Shouldice, S.R.,Vazirani, M.,Headey, S.J.,Plumb, B.R.,Martin, J.L.,Heras, B.,Simpson, J.S.,Scanlon, M.J.
Application of Fragment-Based Screening to the Design of Inhibitors of Escherichia coli DsbA.
Angew.Chem.Int.Ed.Engl., 54:2179-2184, 2015
Cited by
PubMed: 25556635
DOI: 10.1002/anie.201410341
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (1.45 Å)
Structure validation

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