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4U5J

C-Src in complex with Ruxolitinib

Summary for 4U5J
Entry DOI10.2210/pdb4u5j/pdb
DescriptorProto-oncogene tyrosine-protein kinase Src, (3R)-3-cyclopentyl-3-[4-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)-1H-pyrazol-1-yl]propanenitrile (3 entities in total)
Functional Keywordsc-src, ruxolitinib, kinase, inhibitor, transferase-transferase inhibitor complex, transferase/transferase inhibitor
Biological sourceGallus gallus (Chicken)
Cellular locationCell membrane : P00523
Total number of polymer chains2
Total formula weight66066.02
Authors
Chen, Y.,Duan, Y.,Chen, L. (deposition date: 2014-07-25, release date: 2014-09-17, Last modification date: 2022-03-23)
Primary citationDuan, Y.,Chen, L.,Chen, Y.,Fan, X.G.
c-Src Binds to the Cancer Drug Ruxolitinib with an Active Conformation
Plos One, 9:e106225-e106225, 2014
Cited by
PubMed: 25197973
DOI: 10.1371/journal.pone.0106225
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (2.26 Å)
Structure validation

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