4GV7
Human ARTD1 (PARP1) - Catalytic domain in complex with inhibitor ME0328
Summary for 4GV7
Entry DOI | 10.2210/pdb4gv7/pdb |
Descriptor | Poly [ADP-ribose] polymerase 1, 2-methylquinazolin-4(3H)-one (2 entities in total) |
Functional Keywords | nad, adp-ribose, parp1, artd1, artd transferase domain, adp-ribosylation, transferase-transferase inhibitor complex, adp-ribose transferase, transferase/transferase inhibitor |
Biological source | Homo sapiens (human) |
Cellular location | Nucleus: P09874 |
Total number of polymer chains | 4 |
Total formula weight | 161440.49 |
Authors | Karlberg, T.,Thorsell, A.G.,Lindgren, A.E.G.,Ekblad, T.,Spjut, S.,Andersson, C.D.,Weigelt, J.,Linusson, A.,Elofsson, M.,Schuler, H. (deposition date: 2012-08-30, release date: 2013-06-19, Last modification date: 2023-11-08) |
Primary citation | Lindgren, A.E.G.,Karlberg, T.,Thorsell, A.G.,Hesse, M.,Spjut, S.,Ekblad, T.,Andersson, C.D.,Pinto, A.F.,Weigelt, J.,Hottiger, M.O.,Linusson, A.,Elofsson, M.,Schuler, H. PARP Inhibitor with Selectivity Toward ADP-Ribosyltransferase ARTD3/PARP3 Acs Chem.Biol., 8:1698-1703, 2013 Cited by PubMed: 23742272DOI: 10.1021/cb4002014 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.89 Å) |
Structure validation
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