4EH3
Human p38 MAP kinase in complex with NP-F2 and RL87
Summary for 4EH3
Entry DOI | 10.2210/pdb4eh3/pdb |
Related | 4EH2 4EH4 4EH5 4EH6 4EH7 4EH8 4EH9 |
Descriptor | Mitogen-activated protein kinase 14, NARINGENIN, N~4~-cyclopropyl-2-phenylquinazoline-4,7-diamine, ... (4 entities in total) |
Functional Keywords | map kinase insert, kinase-ligand complex, np-fragment, transferase-transferase inhibitor complex, transferase/transferase inhibitor |
Biological source | Homo sapiens (human) |
Cellular location | Cytoplasm: Q16539 |
Total number of polymer chains | 1 |
Total formula weight | 41817.64 |
Authors | Over, B.,Gruetter, C.,Waldmann, H.,Rauh, D. (deposition date: 2012-04-02, release date: 2012-12-05, Last modification date: 2023-09-13) |
Primary citation | Over, B.,Wetzel, S.,Grutter, C.,Nakai, Y.,Renner, S.,Rauh, D.,Waldmann, H. Natural-product-derived fragments for fragment-based ligand discovery. Nat Chem, 5:21-28, 2012 Cited by PubMed: 23247173DOI: 10.1038/nchem.1506 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.4 Å) |
Structure validation
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