3VSP
Human PPAR gamma ligand binding domain in complex with a gamma selective agonist mekt28
Summary for 3VSP
Entry DOI | 10.2210/pdb3vsp/pdb |
Related | 3an3 3VSO |
Descriptor | Peroxisome proliferator-activated receptor gamma, (2R)-2-benzyl-3-[3-({[4-(piperidin-1-yl)benzoyl]amino}methyl)-4-propoxyphenyl]propanoic acid (3 entities in total) |
Functional Keywords | mainly alpha, nuclear receptor, transcription |
Biological source | Homo sapiens (human) |
Cellular location | Nucleus: P37231 |
Total number of polymer chains | 2 |
Total formula weight | 65575.96 |
Authors | Oyama, T.,Waku, T.,Ohashi, M.,Morikawa, K.,Miyachi, H. (deposition date: 2012-04-30, release date: 2013-05-01, Last modification date: 2023-11-08) |
Primary citation | Oyama, T.,Waku, T.,Ohashi, M.,Morikawa, K.,Miyachi, H. Human PPAR gamma ligand binding domain in complex with a gamma selective agonist mekt28 To be Published, |
Experimental method | X-RAY DIFFRACTION (2.4 Å) |
Structure validation
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