3V0P
Crystal structure of the Fucosylgalactoside alpha N-acetylgalactosaminyltransferase (GTA, cisAB mutant L266G, G268A) in complex with a novel UDP-Gal derived inhibitor (4GW) and H-antigen acceptor
3V0P の概要
エントリーDOI | 10.2210/pdb3v0p/pdb |
関連するPDBエントリー | 3IOH 3IOI 3IOJ |
分子名称 | Histo-blood group ABO system transferase, MANGANESE (II) ION, 5-(5-formylthiophen-2-yl)uridine 5'-(trihydrogen diphosphate), ... (6 entities in total) |
機能のキーワード | gta, abo, cisab mutant, rossmann fold, "closed" conformation, glycosyltransferase, glycoprotein, blood group antigen, udp-galnac, metal-binding, manganese, glycosylation, transmembrane, golgi apparatus, secreted, signal-anchor, transferase-transferase inhibitor complex, transferase/transferase inhibitor |
由来する生物種 | Homo sapiens (human) |
細胞内の位置 | Golgi apparatus, Golgi stack membrane; Single-pass type II membrane protein: P16442 |
タンパク質・核酸の鎖数 | 2 |
化学式量合計 | 71419.57 |
構造登録者 | |
主引用文献 | Jrgensen, R.,Pesnot, T.,Lee, H.J.,Palcic, M.M.,Wagner, G.K. Base-modified Donor Analogues Reveal Novel Dynamic Features of a Glycosyltransferase. J.Biol.Chem., 288:26201-26208, 2013 Cited by PubMed: 23836908DOI: 10.1074/jbc.M113.465963 主引用文献が同じPDBエントリー |
実験手法 | X-RAY DIFFRACTION (1.9 Å) |
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