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3RME

AMCase in complex with Compound 5

Summary for 3RME
Entry DOI10.2210/pdb3rme/pdb
Related3RM4 3RM8 3RM9
DescriptorAcidic mammalian chitinase, GLYCEROL, N-ethyl-2-(4-methylpiperazin-1-yl)pyridine-3-carboxamide, ... (4 entities in total)
Functional Keywordshydrolase-hydrolase inhibitor complex, hydrolase/hydrolase inhibitor
Biological sourceHomo sapiens (human)
Cellular locationSecreted. Isoform 2: Cytoplasm. Isoform 3: Cytoplasm: Q9BZP6
Total number of polymer chains2
Total formula weight89087.58
Authors
Olland, A. (deposition date: 2011-04-20, release date: 2011-08-24)
Primary citationCole, D.C.,Olland, A.M.,Jacob, J.,Brooks, J.,Bursavich, M.G.,Czerwinski, R.,Declercq, C.,Johnson, M.,Joseph-McCarthy, D.,Ellingboe, J.W.,Lin, L.,Nowak, P.,Presman, E.,Strand, J.,Tam, A.,Williams, C.M.M.,Yao, S.,Tsao, D.H.H.,Fitz, L.J.
Identification and Characterization of Acidic Mammalian Chitinase Inhibitors
J.Med.Chem., 53:6122-6128, 2010
Cited by
PubMed: 20666458
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (1.8 Å)
Structure validation

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