3RIE
The structure of Plasmodium falciparum spermidine synthase in complex with 5'-methylthioadenosine and N-(3-aminopropyl)-trans-cyclohexane-1,4-diamine
Summary for 3RIE
Entry DOI | 10.2210/pdb3rie/pdb |
Descriptor | Spermidine synthase, 5'-DEOXY-5'-METHYLTHIOADENOSINE, trans-N-(3-aminopropyl)cyclohexane-1,4-diamine, ... (6 entities in total) |
Functional Keywords | rossmann-like fold, rossmann fold, spermidine synthesis, aminopropyl transferase, transferase-transferase inhibitor complex, transferase/transferase inhibitor |
Biological source | Plasmodium falciparum |
Total number of polymer chains | 3 |
Total formula weight | 98597.89 |
Authors | Williams, M.,Sprenger, J.,Persson, L.,Louw, A.I.,Birkholtz, L.,Al-Karadaghi, S. (deposition date: 2011-04-13, release date: 2012-04-25, Last modification date: 2023-09-13) |
Primary citation | Burger, P.B.,Williams, M.,Sprenger, J.,Reeksting, S.B.,Botha, M.,Muller, I.B.,Joubert, F.,Birkholtz, L.M.,Louw, A.I. A novel inhibitor of Plasmodium falciparum spermidine synthase: a twist in the tail. Malar J, 14:54-54, 2015 Cited by PubMed: 25651815DOI: 10.1186/s12936-015-0572-z PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (1.9 Å) |
Structure validation
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