3MY1
Structure of CDK9/cyclinT1 in complex with DRB
Summary for 3MY1
Entry DOI | 10.2210/pdb3my1/pdb |
Related | 3BLH 3BLQ 3BLR 3MY5 |
Descriptor | Cell division protein kinase 9, Cyclin-T1, PHOSPHATE ION, ... (6 entities in total) |
Functional Keywords | cdk-cyclin complex, phosphorylated, transcription-protein binding-inhibitor complex, transcription/protein binding/inhibitor |
Biological source | Homo sapiens (human) More |
Cellular location | Nucleus: P50750 O60563 |
Total number of polymer chains | 2 |
Total formula weight | 69048.09 |
Authors | Baumli, S.,Johnson, L.N. (deposition date: 2010-05-09, release date: 2010-09-29, Last modification date: 2023-11-01) |
Primary citation | Baumli, S.,Endicott, J.A.,Johnson, L.N. Halogen bonds form the basis for selective P-TEFb inhibition by DRB Chem.Biol., 17:931-936, 2010 Cited by PubMed: 20851342DOI: 10.1016/j.chembiol.2010.07.012 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.8 Å) |
Structure validation
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