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3MHU

Crystal structure of dihydroorotate dehydrogenase from Leishmania major in complex with 5-Nitroorotic acid

Summary for 3MHU
Entry DOI10.2210/pdb3mhu/pdb
Related3C3N 3GYE
DescriptorDihydroorotate dehydrogenase, FLAVIN MONONUCLEOTIDE, 5-nitro-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxylic acid, ... (6 entities in total)
Functional Keywordsdihydroorotate dehydrogenase, pyrd, oxidoreductase
Biological sourceLeishmania major
Total number of polymer chains2
Total formula weight76552.85
Authors
Pinheiro, M.P.,Rocha, J.R.,Cheleski, J.,Montanari, C.A.,Nonato, M.C. (deposition date: 2010-04-08, release date: 2011-02-23, Last modification date: 2023-09-06)
Primary citationCheleski, J.,Rocha, J.R.,Pinheiro, M.P.,Wiggers, H.J.,da Silva, A.B.,Nonato, M.C.,Montanari, C.A.
Novel insights for dihydroorotate dehydrogenase class 1A inhibitors discovery.
Eur.J.Med.Chem., 45:5899-5909, 2010
Cited by
PubMed: 20965617
DOI: 10.1016/j.ejmech.2010.09.055
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (1.85 Å)
Structure validation

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