3KGC
Isolated ligand binding domain dimer of GluA2 ionotropic glutamate receptor in complex with glutamate, LY 404187 and ZK 200775
Summary for 3KGC
Entry DOI | 10.2210/pdb3kgc/pdb |
Related | 3KG2 |
Descriptor | Glutamate receptor 2, GLUTAMIC ACID, SULFATE ION, ... (6 entities in total) |
Functional Keywords | glutamate receptor, s1s2, agonist, antagonist, modulator, soluble domain, ligand binding, ion transport, ionic channel, postsynaptic cell membrane, receptor, synapse, membrane protein, glutamate, ly 404187, zk 200775, transport protein |
Biological source | Rattus norvegicus (rat) More |
Total number of polymer chains | 2 |
Total formula weight | 59480.28 |
Authors | Sobolevsky, A.I.,Rosconi, M.P.,Gouaux, E. (deposition date: 2009-10-28, release date: 2009-12-15, Last modification date: 2023-09-06) |
Primary citation | Sobolevsky, A.I.,Rosconi, M.P.,Gouaux, E. X-ray structure, symmetry and mechanism of an AMPA-subtype glutamate receptor Nature, 462:745-755, 2009 Cited by PubMed: 19946266PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (1.55 Å) |
Structure validation
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