3FUR
Crystal Structure of PPARg in complex with INT131
Summary for 3FUR
Entry DOI | 10.2210/pdb3fur/pdb |
Descriptor | Peroxisome proliferator-activated receptor gamma, Nuclear receptor coactivator 1, 2,4-dichloro-N-[3,5-dichloro-4-(quinolin-3-yloxy)phenyl]benzenesulfonamide, ... (5 entities in total) |
Functional Keywords | nuclear receptor, ppargamma, partial agonist, activator, alternative splicing, diabetes mellitus, disease mutation, dna-binding, metal-binding, nucleus, obesity, phosphoprotein, polymorphism, receptor, transcription, transcription regulation, zinc, zinc-finger, int131, transcription-transcription regulator complex, transcription/transcription regulator |
Biological source | Homo sapiens (Human) More |
Total number of polymer chains | 2 |
Total formula weight | 32987.36 |
Authors | Wang, Z.,Liu, J.,Walker, N. (deposition date: 2009-01-14, release date: 2009-06-09, Last modification date: 2024-03-20) |
Primary citation | Motani, A.,Wang, Z.,Weiszmann, J.,McGee, L.R.,Lee, G.,Liu, Q.,Staunton, J.,Fang, Z.,Fuentes, H.,Lindstrom, M.,Liu, J.,Biermann, D.H.,Jaen, J.,Walker, N.P.,Learned, R.M.,Chen, J.L.,Li, Y. INT131: a selective modulator of PPAR gamma. J.Mol.Biol., 386:1301-1311, 2009 Cited by PubMed: 19452630DOI: 10.1016/j.jmb.2009.01.025 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.3 Å) |
Structure validation
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