3EE5
Crystal structure of human M340H-Beta1,4-Galactosyltransferase-I (M340H-B4GAL-T1) in complex with GLCNAC-Beta1,3-Gal-Beta-Naphthalenemethanol
Summary for 3EE5
Entry DOI | 10.2210/pdb3ee5/pdb |
Related | 2AEC |
Descriptor | Beta-1,4-galactosyltransferase 1, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-3)-beta-D-galactopyranose, 6-AMINOHEXYL-URIDINE-C1,5'-DIPHOSPHATE, ... (10 entities in total) |
Functional Keywords | closed conformation, carbohydrate acceptor binding, alternative initiation, cell membrane, congenital disorder of glycosylation, glycoprotein, glycosyltransferase, golgi apparatus, manganese, membrane, metal-binding, secreted, signal-anchor, transferase, transmembrane |
Biological source | Homo sapiens (Human) |
Total number of polymer chains | 3 |
Total formula weight | 103892.03 |
Authors | Ramakrishnan, B.,Qasba, P.K. (deposition date: 2008-09-04, release date: 2009-01-06, Last modification date: 2023-08-30) |
Primary citation | Brown, J.R.,Yang, F.,Sinha, A.,Ramakrishnan, B.,Tor, Y.,Qasba, P.K.,Esko, J.D. Deoxygenated Disaccharide Analogs as Specific Inhibitors of {beta}1-4-Galactosyltransferase 1 and Selectin-mediated Tumor Metastasis J.Biol.Chem., 284:4952-4959, 2009 Cited by PubMed: 19106107DOI: 10.1074/jbc.M805782200 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.2 Å) |
Structure validation
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