3D20
Crystal structure of HIV-1 mutant I54V and inhibitor DARUNAVIA
3D20 の概要
エントリーDOI | 10.2210/pdb3d20/pdb |
関連するPDBエントリー | 3CYW 3CYX 3D1X 3D1Y 3D1Z |
分子名称 | HIV-1 Protease, SODIUM ION, CHLORIDE ION, ... (5 entities in total) |
機能のキーワード | drug resistance; hiv-1, i54v, flap mutant, aids, aspartyl protease, capsid maturation, capsid protein, dna integration, dna recombination, dna-directed dna polymerase, endonuclease, hydrolase, lipoprotein, magnesium, membrane, metal-binding, multifunctional enzyme, myristate, nuclease, nucleotidyltransferase, nucleus, phosphoprotein, protease, rna-binding, rna-directed dna polymerase, transferase, viral nucleoprotein, virion, zinc-finger |
由来する生物種 | Human immunodeficiency virus type 1 (HIV-1) |
細胞内の位置 | Matrix protein p17: Virion (Potential). Capsid protein p24: Virion (Potential). Nucleocapsid protein p7: Virion (Potential). Reverse transcriptase/ribonuclease H: Virion (Potential). Integrase: Virion (Potential): P04587 |
タンパク質・核酸の鎖数 | 2 |
化学式量合計 | 22094.86 |
構造登録者 | Liu, F.,Kovalesky, A.Y.,Tie, Y.,Ghosh, A.K.,Harrison, R.W.,Weber, I.T. (登録日: 2008-05-07, 公開日: 2008-05-27, 最終更新日: 2023-08-30) |
主引用文献 | Liu, F.,Kovalevsky, A.Y.,Tie, Y.,Ghosh, A.K.,Harrison, R.W.,Weber, I.T. Effect of flap mutations on structure of HIV-1 protease and inhibition by saquinavir and darunavir. J.Mol.Biol., 381:102-115, 2008 Cited by PubMed: 18597780DOI: 10.1016/j.jmb.2008.05.062 主引用文献が同じPDBエントリー |
実験手法 | X-RAY DIFFRACTION (1.05 Å) |
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