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2ZVT

Cys285Ser mutant PPARgamma ligand-binding domain complexed with 15-deoxy-delta12,14-prostaglandin J2

Summary for 2ZVT
Entry DOI10.2210/pdb2zvt/pdb
Related2ZK1
DescriptorPeroxisome proliferator-activated receptor gamma, (5E,14E)-11-oxoprosta-5,9,12,14-tetraen-1-oic acid (3 entities in total)
Functional Keywordsanti parallel helix sandwich, activator, alternative splicing, diabetes mellitus, disease mutation, dna-binding, metal-binding, nucleus, obesity, phosphoprotein, polymorphism, receptor, transcription, transcription regulation, zinc, zinc-finger
Biological sourceHomo sapiens (human)
Cellular locationNucleus: P37231
Total number of polymer chains2
Total formula weight65662.04
Authors
Waku, T.,Oyama, T.,Shiraki, T.,Morikawa, K. (deposition date: 2008-11-19, release date: 2009-10-06, Last modification date: 2023-11-01)
Primary citationWaku, T.,Shiraki, T.,Oyama, T.,Morikawa, K.
Atomic structure of mutant PPARgamma LBD complexed with 15d-PGJ2: novel modulation mechanism of PPARgamma/RXRalpha function by covalently bound ligands
Febs Lett., 583:320-324, 2009
Cited by
PubMed: 19101554
DOI: 10.1016/j.febslet.2008.12.017
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (1.9 Å)
Structure validation

217705

數據於2024-03-27公開中

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