2XR9
Crystal structure of Autotaxin (ENPP2)
Summary for 2XR9
Entry DOI | 10.2210/pdb2xr9/pdb |
Related | 2XRG |
Descriptor | ECTONUCLEOTIDE PYROPHOSPHATASE/PHOSPHODIESTERASE FAMILY MEMBER 2, beta-D-mannopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, THIOCYANATE ION, ... (8 entities in total) |
Functional Keywords | hydrolase, lysophosphatidylcholine, somatomedin, inflammation, metastasis, neuropathic pain, vascular development, neural development |
Biological source | RATTUS NORVEGICUS (NORWAY RAT) |
Total number of polymer chains | 1 |
Total formula weight | 99684.71 |
Authors | Kamtekar, S.,Hausmann, J.,Day, J.E.,Christodoulou, E.,Perrakis, A. (deposition date: 2010-09-13, release date: 2011-01-19, Last modification date: 2023-12-20) |
Primary citation | Hausmann, J.,Kamtekar, S.,Christodoulou, E.,Day, J.E.,Wu, T.,Fulkerson, Z.,Albers, H.M.,van Meeteren, L.A.,Houben, A.J.,van Zeijl, L.,Jansen, S.,Andries, M.,Hall, T.,Pegg, L.E.,Benson, T.E.,Kasiem, M.,Harlos, K.,Kooi, C.W.,Smyth, S.S.,Ovaa, H.,Bollen, M.,Morris, A.J.,Moolenaar, W.H.,Perrakis, A. Structural basis of substrate discrimination and integrin binding by autotaxin. Nat. Struct. Mol. Biol., 18:198-204, 2011 Cited by PubMed: 21240271DOI: 10.1038/nsmb.1980 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.05 Å) |
Structure validation
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