2XEI
Human glutamate carboxypeptidase II in complex with Antibody- Recruiting Molecule ARM-P2
Summary for 2XEI
Entry DOI | 10.2210/pdb2xei/pdb |
Related | 1Z8L 2C6C 2C6G 2C6P 2CIJ 2JBJ 2JBK 2XEF 2XEG 2XEJ |
Descriptor | GLUTAMATE CARBOXYPEPTIDASE 2, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, alpha-D-mannopyranose-(1-3)-beta-D-mannopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ... (9 entities in total) |
Functional Keywords | metallopeptidase, hydrolase |
Biological source | HOMO SAPIENS (HUMAN) |
Cellular location | Cell membrane ; Single-pass type II membrane protein . Isoform PSMA': Cytoplasm: Q04609 |
Total number of polymer chains | 1 |
Total formula weight | 83407.49 |
Authors | Zhang, A.X.,Murelli, R.P.,Barinka, C.,Michel, J.,Cocleaza, A.,Jorgensen, W.L.,Lubkowski, J.,Spiegel, D.A. (deposition date: 2010-05-14, release date: 2010-09-08, Last modification date: 2023-12-20) |
Primary citation | Zhang, A.X.,Murelli, R.P.,Barinka, C.,Michel, J.,Cocleaza, A.,Jorgensen, W.L.,Lubkowski, J.,Spiegel, D.A. A Remote Arene-Binding Site on Prostate Specific Membrane Antigen Revealed by Antibody-Recruiting Small Molecules. J.Am.Chem.Soc., 132:12711-, 2010 Cited by PubMed: 20726553DOI: 10.1021/JA104591M PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (1.69 Å) |
Structure validation
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