2VRX
Structure of Aurora B kinase in complex with ZM447439
Summary for 2VRX
Entry DOI | 10.2210/pdb2vrx/pdb |
Related | 2BFX 2BFY 2VGO 2VGP |
Descriptor | SERINE/THREONINE-PROTEIN KINASE 12-A, INNER CENTROMERE PROTEIN A, N-(4-{[6-methoxy-7-(3-morpholin-4-ylpropoxy)quinazolin-4-yl]amino}phenyl)benzamide, ... (4 entities in total) |
Functional Keywords | serine/threonine-protein kinase, kinase, nucleus, mitosis, magnesium, cell cycle/transferase, centromere, microtubule, atp-binding, transferase, anti-cancer drug target, phosphoprotein, protein kinase, nucleotide-binding, coiled coil, cell division, metal-binding, cell cycle-transferase complex |
Biological source | XENOPUS LAEVIS (AFRICAN CLAWED FROG) More |
Cellular location | Nucleus: Q6DE08 Chromosome, centromere: O13024 |
Total number of polymer chains | 4 |
Total formula weight | 78284.39 |
Authors | Girdler, F.,Sessa, F.,Patercoli, S.,Villa, F.,Ridgway, E.,Musacchio, A.,Taylor, S.S. (deposition date: 2008-04-16, release date: 2008-07-01, Last modification date: 2011-07-13) |
Primary citation | Girdler, F.,Sessa, F.,Patercoli, S.,Villa, F.,Musacchio, A.,Taylor, S.S. Molecular Basis of Drug Resistance in Aurora Kinases. Chem.Biol., 15:552-, 2008 Cited by PubMed: 18559266DOI: 10.1016/J.CHEMBIOL.2008.04.013 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (1.86 Å) |
Structure validation
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