2PZI
Crystal Structure of Protein kinase PknG from Mycobacterium tuberculosis in Complex with Tetrahydrobenzothiophene AX20017
Summary for 2PZI
Entry DOI | 10.2210/pdb2pzi/pdb |
Related | 1ATP 1O6Y 2FUM |
Descriptor | Probable serine/threonine-protein kinase pknG, CHLORIDE ION, CADMIUM ION, ... (6 entities in total) |
Functional Keywords | serine/threonine-protein kinase, atp-recognition, kinase-inhibitor complex, rubredoxin fold, tpr domain, transferase |
Biological source | Mycobacterium tuberculosis |
Total number of polymer chains | 2 |
Total formula weight | 149707.49 |
Authors | Honnappa, S.,Steinmetz, M.O. (deposition date: 2007-05-18, release date: 2007-07-24, Last modification date: 2024-02-21) |
Primary citation | Scherr, N.,Honnappa, S.,Kunz, G.,Mueller, P.,Jayachandran, R.,Winkler, F.,Pieters, J.,Steinmetz, M.O. Structural basis for the specific inhibition of protein kinase G, a virulence factor of Mycobacterium tuberculosis. Proc.Natl.Acad.Sci.Usa, 104:12151-12156, 2007 Cited by PubMed: 17616581DOI: 10.1073/pnas.0702842104 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.4 Å) |
Structure validation
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