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2JKQ

Focal Adhesion Kinase catalytic domain in complex with bis-anilino pyrimidine inhibitor

Summary for 2JKQ
Entry DOI10.2210/pdb2jkq/pdb
Related1KTM 1PV3 1QVX 2AEH 2AL6 2J0J 2J0K 2J0L 2J0M 2JKK 2JKM 2JKO
DescriptorFOCAL ADHESION KINASE 1, 4-(1,4'-bipiperidin-1'-yl)-7-({5-chloro-2-[(2-methoxyphenyl)amino]pyrimidin-4-yl}amino)-2-methyl-2,3-dihydro-1H-isoindol-1-one (3 entities in total)
Functional Keywordstransferase, nucleotide-binding, tyrosine-protein kinase, kinase inhibitor, integrin signaling, kinase, atp-binding, cell migration, focal adhesion
Biological sourceGALLUS GALLUS (CHICKEN)
Total number of polymer chains1
Total formula weight32320.87
Authors
Lietha, D.,Eck, M.J. (deposition date: 2008-08-29, release date: 2008-09-09, Last modification date: 2023-12-13)
Primary citationLietha, D.,Eck, M.J.
Crystal Structures of the Fak Kinase in Complex with Tae226 and Related Bis-Anilino Pyrimidine Inhibitors Reveal a Helical Dfg Conformation.
Plos One, 3:E3800-, 2008
Cited by
PubMed: 19030106
DOI: 10.1371/JOURNAL.PONE.0003800
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (2.6 Å)
Structure validation

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