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2EXC

Inhibitor complex of JNK3

Summary for 2EXC
Entry DOI10.2210/pdb2exc/pdb
DescriptorMitogen-activated protein kinase 10, N-{2'-[(4-FLUOROPHENYL)AMINO]-4,4'-BIPYRIDIN-2-YL}-4-METHOXYCYCLOHEXANECARBOXAMIDE (3 entities in total)
Functional Keywordsenzyme-inhibitor complex, kinase inhibitor, transferase
Biological sourceHomo sapiens (human)
Cellular locationCytoplasm: P53779
Total number of polymer chains1
Total formula weight41601.12
Authors
Xue, Y. (deposition date: 2005-11-08, release date: 2006-11-14, Last modification date: 2024-02-14)
Primary citationSwahn, B.-M.,Xue, Y.,Arzel, E.,Kallin, E.,Magnus, A.,Plobeck, N.,Viklund, J.
Inhibitor complex of JNK3
To be Published,
Experimental method
X-RAY DIFFRACTION (2.75 Å)
Structure validation

218853

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