22HA

The crystal structure of BRD4-BD1 in complex with inhibitor C2

This is a non-PDB format compatible entry.

Summary for 22HA

• Entry DOI: 10.2210/pdb22ha/pdb
• Descriptor: Bromodomain-containing protein 4, 3-chloranyl-~{N}-(3,4-dimethoxyphenyl)-4-[[(1~{R},2~{S})-2-methyl-3-oxidanylidene-cyclopentyl]amino]benzamide (3 entities in total)
• Functional Keywords: brd4, bd1, inhibitor, structural protein
• Biological source: Homo sapiens (human)
• Total number of polymer chains: 1
• Total formula weight: 15688.93

Authors

Wu, C.Y.,Zhang, J.F. (deposition date: 2026-01-10, release date: 2026-09-23)

• Primary citation: Wu, C.Y.,Zhang, J.F.; The crystal structure of BRD4-BD1 in complex with C2; To Be Published,

Experimental method

X-RAY DIFFRACTION (2.1 Å)