1RPW
Crystal Structure Of The Multidrug Binding Protein Qacr Bound To The Diamidine Hexamidine
Summary for 1RPW
Entry DOI | 10.2210/pdb1rpw/pdb |
Related | 1JT6 1JTY 1JUS |
Descriptor | Transcriptional regulator qacR, SULFATE ION, 4,4'[1,6-HEXANEDIYLBIS(OXY)]BISBENZENECARBOXIMIDAMIDE, ... (4 entities in total) |
Functional Keywords | qacr hexamidine, transcription |
Biological source | Staphylococcus aureus |
Total number of polymer chains | 4 |
Total formula weight | 90892.28 |
Authors | Murray, D.S.,Schumacher, M.A.,Brennan, R.G. (deposition date: 2003-12-03, release date: 2004-06-01, Last modification date: 2023-08-23) |
Primary citation | Murray, D.S.,Schumacher, M.A.,Brennan, R.G. Crystal structures of QacR-diamidine complexes reveal additional multidrug-binding modes and a novel mechanism of drug charge neutralization. J.Biol.Chem., 279:14365-14371, 2004 Cited by PubMed: 14726520DOI: 10.1074/jbc.M313870200 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.9 Å) |
Structure validation
Download full validation report