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1E8X

STRUCTURAL INSIGHTS INTO PHOSHOINOSITIDE 3-KINASE ENZYMATIC MECHANISM AND SIGNALLING

Replaces:  1QMM
Summary for 1E8X
Entry DOI10.2210/pdb1e8x/pdb
Related1E7U 1E7V 1E8W 1QMM
DescriptorPHOSPHATIDYLINOSITOL 3-KINASE CATALYTIC SUBUNIT, ADENOSINE-5'-TRIPHOSPHATE, LUTETIUM (III) ION, ... (4 entities in total)
Functional Keywordsphosphoinositide 3-kinase gamma, secondary messenger generation, pi3k, pi 3k
Biological sourceSUS SCROFA (WILD BOAR)
Total number of polymer chains1
Total formula weight112034.44
Authors
Walker, E.H.,Perisic, O.,Ried, C.,Stephens, L.,Williams, R.L. (deposition date: 2000-10-03, release date: 2000-10-26, Last modification date: 2018-10-24)
Primary citationWalker, E.H.,Pacold, M.E.,Perisic, O.,Stephens, L.,Hawkins, P.T.,Whymann, M.P.,Williams, R.L.
Structural Determinations of Phosphoinositide 3-Kinase Inhibition by Wortmannin, Ly294002, Quercetin, Myricetin and Staurosporine
Mol.Cell, 6:909-, 2000
Cited by
PubMed: 11090628
DOI: 10.1016/S1097-2765(05)00089-4
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (2.2 Å)
Structure validation

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