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1P45

Targeting tuberculosis and malaria through inhibition of enoyl reductase: compound activity and structural data

Summary for 1P45
Entry DOI10.2210/pdb1p45/pdb
Related1P44
DescriptorEnoyl-[acyl-carrier-protein] reductase [NADH], NICOTINAMIDE-ADENINE-DINUCLEOTIDE, TRICLOSAN, ... (4 entities in total)
Functional Keywordsinha, short chain dehydrogenase reductase, triclosan, rossmann fold, enoyl-acp reductase, structural genomics, psi, protein structure initiative, tb structural genomics consortium, tbsgc, oxidoreductase
Biological sourceMycobacterium tuberculosis
Total number of polymer chains2
Total formula weight59305.04
Authors
Primary citationKuo, M.R.,Morbidoni, H.R.,Alland, D.,Sneddon, S.F.,Gourlie, B.B.,Staveski, M.M.,Leonard, M.,Gregory, J.S.,Janjigian, A.D.,Yee, C.,Musser, J.M.,Kreiswirth, B.,Iwamoto, H.,Perozzo, R.,Jacobs, W.R.,Sacchettini, J.C.,Fidock, D.A.
Targeting tuberculosis and malaria through inhibition of Enoyl reductase: compound activity and structural data.
J.Biol.Chem., 278:20851-20859, 2003
Cited by
PubMed: 12606558
DOI: 10.1074/jbc.M211968200
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (2.6 Å)
Structure validation

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