1JCS
CRYSTAL STRUCTURE OF RAT PROTEIN FARNESYLTRANSFERASE COMPLEXED WITH THE PEPTIDE SUBSTRATE TKCVFM AND AN ANALOG OF FARNESYL DIPHOSPHATE
1JCS の概要
エントリーDOI | 10.2210/pdb1jcs/pdb |
関連するPDBエントリー | 1D8D 1FT1 1JCQ 1JCR |
分子名称 | PROTEIN FARNESYLTRANSFERASE, ALPHA SUBUNIT, PROTEIN FARNESYLTRANSFERASE, BETA SUBUNIT, SYNTHETIC HEXAPEPTIDE TKCVFM, ... (7 entities in total) |
機能のキーワード | ftase, pft, pftase, ft, fpt, farnesyltransferase, farnesyl transferase, farnesyl protein transferase, caax, ras, cancer, inhibitor, transferase, transferase-transferase inhibitor complex, transferase/transferase inhibitor |
由来する生物種 | Rattus norvegicus (Norway rat) 詳細 |
タンパク質・核酸の鎖数 | 3 |
化学式量合計 | 94094.28 |
構造登録者 | |
主引用文献 | Long, S.B.,Hancock, P.J.,Kral, A.M.,Hellinga, H.W.,Beese, L.S. The crystal structure of human protein farnesyltransferase reveals the basis for inhibition by CaaX tetrapeptides and their mimetics. Proc.Natl.Acad.Sci.USA, 98:12948-12953, 2001 Cited by PubMed: 11687658DOI: 10.1073/pnas.241407898 主引用文献が同じPDBエントリー |
実験手法 | X-RAY DIFFRACTION (2.2 Å) |
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