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1TYE

Structural basis for allostery in integrins and binding of ligand-mimetic therapeutics to the platelet receptor for fibrinogen

Summary for 1TYE
Entry DOI10.2210/pdb1tye/pdb
Related1TXV 1TY3 1TY5 1TY6 1TY7
DescriptorIntegrin alpha-IIb, Integrin beta-3, beta-D-mannopyranose-(1-3)-alpha-D-mannopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ... (9 entities in total)
Functional Keywordscrystal structure; platelet integrin alphaiibbeta3; fibrinogen binding; allostery; therapeutic antagonism, cell adhesion
Biological sourceHomo sapiens (human)
More
Total number of polymer chains6
Total formula weight298452.84
Authors
Xiao, T.,Takagi, J.,Coller, B.S.,Wang, J.-H.,Springer, T.A. (deposition date: 2004-07-07, release date: 2004-10-12, Last modification date: 2023-08-23)
Primary citationXiao, T.,Takagi, J.,Coller, B.S.,Wang, J.-H.,Springer, T.A.
Structural basis for allostery in integrins and binding to fibrinogen-mimetic therapeutics
Nature, 432:59-67, 2004
Cited by
PubMed: 15378069
DOI: 10.1038/nature02976
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (2.9 Å)
Structure validation

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