1QR3
Structure of porcine pancreatic elastase in complex with FR901277, a novel macrocyclic inhibitor of elastases at 1.6 angstrom resolution
Summary for 1QR3
Entry DOI | 10.2210/pdb1qr3/pdb |
Related PRD ID | PRD_000561 |
Descriptor | Chymotrypsin-like elastase family member 1, FR901277 Inhibitor, CALCIUM ION, ... (5 entities in total) |
Functional Keywords | protease, hydrolase-hydrolase inhibitor complex, hydrolase/hydrolase inhibitor |
Biological source | Sus scrofa (Pig) More |
Total number of polymer chains | 2 |
Total formula weight | 27080.27 |
Authors | Nakanishi, I.,Kinoshita, T.,Sato, A.,Tada, T. (deposition date: 1999-06-18, release date: 2000-06-21, Last modification date: 2023-11-15) |
Primary citation | Nakanishi, I.,Kinoshita, T.,Sato, A.,Tada, T. Structure of porcine pancreatic elastase complexed with FR901277, a novel macrocyclic inhibitor of elastases, at 1.6 A resolution. Biopolymers, 53:434-445, 2000 Cited by PubMed: 10738204DOI: 10.1002/(SICI)1097-0282(20000415)53:5<434::AID-BIP7>3.0.CO;2-5 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (1.6 Å) |
Structure validation
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