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9MX2

Human G protein-coupled receptor kinase 5-D311N in complex with sangivamycin soaked in pH 6

Entity
Entity IDChain IDDescriptionTypeChain lengthFormula weightNumber of moleculesDB Name (Accession)Biological sourceDescriptive keywords
1A
(A)
G protein-coupled receptor kinase 5polymer59968957.81UniProt (P34947)
Pfam (PF00615)
Pfam (PF00069)
Homo sapiens (human)G protein-coupled receptor kinase GRK5
2B
(A)
SANGIVAMYCINnon-polymer309.31Chemie (SGV)
PubChem (16760643)
PubChem (5153)
PubChem (14978)
PubChem (44330426)
PubChem (57685061)
PubChem (46875748)
PubChem (70829033)
PubChem (3007220)
PubChem (89687375)
PubChem (92209899)
PubChem (92209900)
PubChem (92209901)
PubChem (6712998)
PubChem (101037982)
PubChem (10403057)
PubChem (10448038)
PubChem (142650208)
PubChem (162968206)
3C
(A)
POTASSIUM IONnon-polymer39.11Chemie (K)
PubChem (813)
Sequence modifications
A: 1 - 590 (UniProt: P34947)
PDBExternal DatabaseDetails
Ace 0-acetylation
Asn 311Asp 311engineered mutation
Val 591-expression tag
Asp 592-expression tag
His 593-expression tag
His 594-expression tag
His 595-expression tag
His 596-expression tag
His 597-expression tag
His 598-expression tag
Sequence viewer
Contents of the asymmetric unit
PolymersNumber of chains1
Total formula weight68957.8
Non-Polymers*Number of molecules2
Total formula weight348.4
All*Total formula weight69306.1
*Water molecules are not included.

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PDB entries from 2026-05-13

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