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9CKO

Human G protein-coupled receptor kinase 5 wild-type in complex with sangivamycin

Entity
Entity IDChain IDDescriptionTypeChain lengthFormula weightNumber of moleculesDB Name (Accession)Biological sourceDescriptive keywords
1A
(A)
G protein-coupled receptor kinase 5polymer59868932.71UniProt (P34947)
Pfam (PF00615)
Pfam (PF00069)
Homo sapiens (human)G protein-coupled receptor kinase GRK5
2B
(A)
ACETYL GROUPnon-polymer44.11Chemie (ACE)
3C
(A)
SANGIVAMYCINnon-polymer309.31Chemie (SGV)
PubChem (5153)
PubChem (14978)
PubChem (6712998)
PubChem (10403057)
PubChem (10448038)
PubChem (16760643)
PubChem (44330426)
PubChem (46875748)
PubChem (3007220)
PubChem (57685061)
PubChem (70829033)
PubChem (89687375)
PubChem (92209899)
PubChem (92209900)
PubChem (92209901)
PubChem (101037982)
PubChem (142650208)
PubChem (162968206)
4D
(A)
POTASSIUM IONnon-polymer39.11Chemie (K)
PubChem (813)
5E
(A)
waterwater18.072Chemie (HOH)
Sequence modifications
A: 1 - 590 (UniProt: P34947)
PDBExternal DatabaseDetails
Val 591-expression tag
Asp 592-expression tag
His 593-expression tag
His 594-expression tag
His 595-expression tag
His 596-expression tag
His 597-expression tag
His 598-expression tag
Sequence viewer
Contents of the asymmetric unit
PolymersNumber of chains1
Total formula weight68932.7
Non-Polymers*Number of molecules3
Total formula weight392.4
All*Total formula weight69325.1
*Water molecules are not included.

251801

PDB entries from 2026-04-08

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