9BJK
Inactive mu opioid receptor bound to Nb6, naloxone and NAM
This is a non-PDB format compatible entry.
Entity
Entity ID | Chain ID | Description | Type | Chain length | Formula weight | Number of molecules | DB Name (Accession) | Biological source | Descriptive keywords |
1 | N | kappa opioid receptor Nanobody 6 | polymer | 133 | 14730.3 | 1 | Lama glama | ||
2 | R | Mu-type opioid receptor | polymer | 426 | 47920.7 | 1 | UniProt (P42866) In PDB | Mus musculus (house mouse) | M-OR-1,MOR-1 |
3 | R | Naloxone | non-polymer | 327.4 | 1 | Chemie (A1APV) | |||
4 | R | Nalpha-[({(1M)-1-[5-(benzyloxy)pyridin-3-yl]naphthalen-2-yl}sulfanyl)acetyl]-3-methoxy-N,4-dimethyl-L-phenylalaninamide | non-polymer | 605.7 | 1 | Chemie (A1APU) |
Sequence modifications
R: 6 - 398 (UniProt: P42866)
PDB | External Database | Details |
---|---|---|
Met -19 | - | initiating methionine |
Lys -18 | - | expression tag |
Thr -17 | - | expression tag |
Ile -16 | - | expression tag |
Ile -15 | - | expression tag |
Ala -14 | - | expression tag |
Leu -13 | - | expression tag |
Ser -12 | - | expression tag |
Tyr -11 | - | expression tag |
Ile -10 | - | expression tag |
Phe -9 | - | expression tag |
Cys -8 | - | expression tag |
Leu -7 | - | expression tag |
Val -6 | - | expression tag |
Phe -5 | - | expression tag |
Ala -4 | - | expression tag |
Asp -3 | - | expression tag |
Tyr -2 | - | expression tag |
Lys -1 | - | expression tag |
Asp 0 | - | expression tag |
Asp 1 | - | expression tag |
Asp 2 | - | expression tag |
Asp 3 | - | expression tag |
Ala 4 | - | expression tag |
Met 5 | - | expression tag |
Leu 264 | Met 264 | engineered mutation |
Arg 269 | Lys 269 | engineered mutation |
Asp 399 | - | expression tag |
Ile 400 | - | expression tag |
His 401 | - | expression tag |
His 402 | - | expression tag |
His 403 | - | expression tag |
His 404 | - | expression tag |
His 405 | - | expression tag |
His 406 | - | expression tag |
Sequence viewer
Contents of the asymmetric unit
Polymers | Number of chains | 2 |
Total formula weight | 62651.0 | |
Non-Polymers* | Number of molecules | 2 |
Total formula weight | 933.1 | |
All* | Total formula weight | 63584.1 |