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9AYL

Cryo-EM structure of human Cav3.2 with ACT-709478

This is a non-PDB format compatible entry.
Entity
Entity IDChain IDDescriptionTypeChain lengthFormula weightNumber of moleculesDB Name (Accession)Biological sourceDescriptive keywords
1A
(A)
Voltage-dependent T-type calcium channel subunit alpha-1Hpolymer2116234853.61UniProt (O95180)
Pfam (PF00520)
Homo sapiens (human)Low-voltage-activated calcium channel alpha1 3.2 subunit,Voltage-gated calcium channel subunit alpha Cav3.2
2B
(A)
N-{1-[(5-cyanopyridin-2-yl)methyl]-1H-pyrazol-3-yl}-2-{4-[1-(trifluoromethyl)cyclopropyl]phenyl}acetamidenon-polymer425.41Chemie (A1AHK)
PubChem (118560618)
3C, D
(A)
2-acetamido-2-deoxy-beta-D-glucopyranosenon-polymer221.22Chemie (NAG)
4E
(A)
CALCIUM IONnon-polymer40.11Chemie (CA)
PubChem (271)
5F
(A)
1-O-OCTADECYL-SN-GLYCERO-3-PHOSPHOCHOLINEnon-polymer510.71Chemie (LPE)
PubChem (3855)
PubChem (9546711)
PubChem (446876)
6G, I, M, N
(A)
CHOLESTEROL HEMISUCCINATEnon-polymer486.74Chemie (Y01)
PubChem (65082)
PubChem (363416)
PubChem (500055)
PubChem (13301926)
PubChem (13301927)
PubChem (16219150)
PubChem (22210610)
PubChem (45489984)
PubChem (57163942)
PubChem (89891013)
PubChem (99567468)
PubChem (124427194)
PubChem (124897021)
PubChem (124897020)
PubChem (10005657)
PubChem (130340716)
PubChem (11969853)
PubChem (137392566)
PubChem (137496323)
PubChem (155804219)
PubChem (169132514)
PubChem (60078761)
PubChem (73440805)
PubChem (99567469)
PubChem (124301053)
PubChem (124302591)
PubChem (124303794)
PubChem (124421343)
PubChem (124427195)
PubChem (124914595)
PubChem (124914596)
PubChem (131705526)
PubChem (137332121)
PubChem (137496357)
PubChem (146157332)
PubChem (154929912)
PubChem (155199678)
PubChem (156327905)
PubChem (156426247)
PubChem (156516588)
PubChem (166979870)
PubChem (167024614)
PubChem (169132513)
PubChem (170117245)
PubChem (172400028)
7H, J, K, L
(A)
[(2~{R})-3-[2-azanylethoxy(oxidanyl)phosphoryl]oxy-2-pentadecanoyloxy-propyl] pentadecanoatenon-polymer663.94Chemie (JL3)
PubChem (9546808)
PubChem (9546807)
Sequence modifications
A: 1 - 771 (UniProt: O95180)
PDBExternal DatabaseDetails
Met -42-expression tag
Ala -41-expression tag
Ser -40-expression tag
Trp -39-expression tag
Ser -38-expression tag
His -37-expression tag
Pro -36-expression tag
Gln -35-expression tag
Phe -34-expression tag
Glu -33-expression tag
Lys -32-expression tag
Gly -31-expression tag
Gly -30-expression tag
Gly -29-expression tag
Ala -28-expression tag
Arg -27-expression tag
Gly -26-expression tag
Gly -25-expression tag
Ser -24-expression tag
Gly -23-expression tag
Gly -22-expression tag
Gly -21-expression tag
Ser -20-expression tag
Trp -19-expression tag
Ser -18-expression tag
His -17-expression tag
Pro -16-expression tag
Gln -15-expression tag
Phe -14-expression tag
Glu -13-expression tag
Lys -12-expression tag
Gly -11-expression tag
Phe -10-expression tag
Asp -9-expression tag
Tyr -8-expression tag
Lys -7-expression tag
Asp -6-expression tag
Asp -5-expression tag
Asp -4-expression tag
Asp -3-expression tag
Lys -2-expression tag
Gly -1-expression tag
Thr 0-expression tag
A: 772 - 2353 (UniProt: O95180)
Sequence viewer
Contents of the asymmetric unit
PolymersNumber of chains1
Total formula weight234853.6
Non-Polymers*Number of molecules13
Total formula weight6021.1
All*Total formula weight240874.7
*Water molecules are not included.

251801

PDB entries from 2026-04-08

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