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8VJ7

GluA2 bound to GYKI-52466 and Glutamate, Inhibited State 2

This is a non-PDB format compatible entry.
Entity
Entity IDChain IDDescriptionTypeChain lengthFormula weightNumber of moleculesDB Name (Accession)Biological sourceDescriptive keywords
1A, B, C, DIsoform Flip of Glutamate receptor 2polymer79789233.04UniProt (P19491)
Pfam (PF01094)
Pfam (PF10613)
Pfam (PF00060)
In PDB
Rattus norvegicus (Norway rat)GluR-2,AMPA-selective glutamate receptor 2,GluR-B,GluR-K2,Glutamate receptor ionotropic,AMPA 2,GluA2
2A, B, C, DGLUTAMIC ACIDnon-polymer147.14Chemie (GLU)
3A, C, D4-[(5S,8R)-8-methyl-6,7,8,9-tetrahydro-2H,5H-[1,3]dioxolo[4,5-h][2,3]benzodiazepin-5-yl]anilinenon-polymer293.34Chemie (A1AB5)
Sequence modifications
A, B, C, D: 10 - 821 (UniProt: P19491)
PDBExternal DatabaseDetails
Glu 241Asn 256conflict
Leu 382Val 397conflict
-Leu 399deletion
-Thr 400deletion
-Glu 401deletion
-Leu 402deletion
-Pro 403deletion
-Ser 404deletion
Glu 384Gly 405conflict
Asp 385Asn 406conflict
Gln 392Asn 413conflict
-Glu 571deletion
-Trp 572deletion
-His 573deletion
-Thr 574deletion
-Glu 575deletion
-Glu 576deletion
-Phe 577deletion
-Glu 578deletion
-Asp 579deletion
-Gly 580deletion
-Arg 581deletion
-Glu 582deletion
-Thr 583deletion
-Gln 584deletion
-Ser 585deletion
Sequence viewer
Contents of the asymmetric unit
PolymersNumber of chains4
Total formula weight356931.8
Non-Polymers*Number of molecules8
Total formula weight1761.8
All*Total formula weight358693.6
*Water molecules are not included.

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PDB entries from 2024-07-31

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