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8HVI

Activation mechanism of GPR132 by compound NOX-6-7

エンティティ
Entity ID鎖名説明種類鎖長化学式量分子数データベース名(アクセス番号)由来する生物種エンティティの一般名
1A
(R)
Soluble cytochrome b562,Probable G-protein coupled receptor 132polymer51057125.31UniProt (P0ABE7)
UniProt (Q9UNW8)
Pfam (PF07361)
Pfam (PF00001)
Escherichia coliCytochrome b-562,G2 accumulation protein
2B
(B)
Guanine nucleotide-binding protein G(i) subunit alpha-1polymer35440445.11UniProt (P63096)
Pfam (PF00503)
Homo sapiens (human)Adenylate cyclase-inhibiting G alpha protein
3C
(C)
Guanine nucleotide-binding protein G(I)/G(S)/G(T) subunit beta-1polymer35839489.21UniProt (P62873)
Pfam (PF00400)
Homo sapiens (human)Transducin beta chain 1
4D
(D)
Guanine nucleotide-binding protein G(I)/G(S)/G(O) subunit gamma-2polymer586375.31UniProt (P59768)
Pfam (PF00631)
Homo sapiens (human)G gamma-I
5E
(H)
scFv16polymer25026610.61Mus musculus
6F
(R)
3-methyl-5-[(4-oxidanylidene-4-phenyl-butanoyl)amino]-1-benzofuran-2-carboxylic acidnon-polymer351.41Chemie (NFI)
配列変更
R: -98 - -5 (UniProt: P0ABE7)
PDB外部データベース詳細
Met -129-initiating methionine
Lys -128-expression tag
Thr -127-expression tag
Ile -126-expression tag
Ile -125-expression tag
Ala -124-expression tag
Leu -123-expression tag
Ser -122-expression tag
Tyr -121-expression tag
Ile -120-expression tag
Phe -119-expression tag
Cys -118-expression tag
Leu -117-expression tag
Val -116-expression tag
Phe -115-expression tag
Ala -114-expression tag
Asp -113-expression tag
Tyr -112-expression tag
Lys -111-expression tag
Asp -110-expression tag
Asp -109-expression tag
Asp -108-expression tag
Asp -107-expression tag
Lys -106-expression tag
Ala -105-expression tag
Asp -104-expression tag
Leu -103-expression tag
Glu -102-expression tag
Asp -101-expression tag
Asn -100-expression tag
Trp -99-expression tag
Ile -4-linker
Gln -3-linker
Lys -2-linker
Tyr -1-linker
Leu 0-linker
R: 1 - 380 (UniProt: Q9UNW8)
B: 1 - 354 (UniProt: P63096)
PDB外部データベース詳細
Ala 203Gly 203conflict
Ser 326Ala 326conflict
C: 2 - 340 (UniProt: P62873)
PDB外部データベース詳細
Met -17-initiating methionine
His -16-expression tag
His -15-expression tag
His -14-expression tag
His -13-expression tag
His -12-expression tag
His -11-expression tag
Leu -10-expression tag
Glu -9-expression tag
Val -8-expression tag
Leu -7-expression tag
Phe -6-expression tag
Gln -5-expression tag
Gly -4-expression tag
Pro -3-expression tag
Gly -2-expression tag
Ser -1-expression tag
Ser 0-expression tag
Gln 1-expression tag
配列ビューア
非対称単位の内容
タンパク質・
核酸鎖
鎖の数5
化学式量合計170045.5
タンパク質・
核酸・
糖鎖以外*
分子数1
化学式量合計351.4
全て*化学式量合計170396.8
*水分子は含んでいません

239803

件を2025-08-06に公開中

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